List of Kinases for Activity Screening
Table – Kinases for Activity Screening
QuickScout™ Kinase Activity Assays
Target Name | Group | Available Services | Source
Carna Category Number |
|||||||
(Mobility Shift Assay, IMAP™) | Pre-selected Panel | |||||||||
ABL(ABL1) | TK | Km bin. | 1mM | Preincubation | TK | 08-001 | ||||
ABL(ABL1)[E255K] | TK | Km_bin. | 1mM | Preincubation | 08-094 | |||||
ABL(ABL1)[T315I] | TK | Km bin. | 1mM | Preincubation | 08-093 | |||||
ACK (TNK2) | TK | Km bin. | 1mM | 08-196 | ||||||
AKT1 | STK | Km bin. | 1mM | Preincubation | STK | 01-101 | ||||
AKT2 | STK | Km bin. | Preincubation | 01-102 | ||||||
AKT3 | STK | Km bin. | Preincubation | 01-103 | ||||||
ALK | TK | Km bin. | 1mM | Preincubation | 08-518 | |||||
ALK[C1156Y] | TK | Km bin. | 1mM | Preincubation | 08-530 | |||||
ALK[F1174L] | TK | Km bin. | 1mM | Preincubation | 08-519 | |||||
ALK[G1202R] | TK | Km bin. | 1mM | Preincubation | 08-544 | |||||
ALK[G1269A] | TK | Km bin. | 1mM | Preincubation | 08-537 | |||||
ALK[L1196M] | TK | Km bin. | 1mM | Preincubation | 08-529 | |||||
ALK[R1275Q] | TK | Km bin. | 1mM | Preincubation | 08-520 | |||||
ALK[T1151_L1152insT] | TK | Km bin. | 1mM | 08-539 | ||||||
AMPKα1/β1/γ1 (PRKAA1/B1/G1) | STK | Km bin. | 1mM | Preincubation | STK | 02-113 | ||||
AMPKα2/β1/γ1 (PRKAA2/B1/G1) | STK | Km bin. | Preincubation | 02-114 | ||||||
ARG (ABL2) | TK | Km bin. | 1mM | Preincubation | 08-102 | |||||
AurA (AURKA) | STK | Km bin. | 1mM | Preincubation | STK | Cell_Cycle | 05-101 | |||
AurA (AURKA)/TPX2 | STK | Km bin. | Preincubation | 05-186 | ||||||
AurB (AURKB)/INCENP | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 05-102 | ||||
AurC (AURKC) | STK | Km bin. | 1mM | Cell Cycle | 05-103 | |||||
AXL | TK | Km bin. | 1mM | 08-107 | ||||||
BLK | TK | Km bin. | 1mM | 08-164 | ||||||
BMX | TK | Km bin. | 1mM | Preincubation | 08-179 | |||||
BRAF | STK | 1mM (Cascade) | MAPK (Cascade) | 09-122 | ||||||
BRAF[V600E] | STK | 1mM (Cascade) | 09-144 | |||||||
BRK (PTK6) | TK | Km bin. | 1mM | 08-165 | ||||||
BRSK1 | STK | Km bin. | 1mM | Preincubation | 02-115 | |||||
BRSK2 | STK | Km bin. | Preincubation | Cell Cycle | 02-116 | |||||
BTK | TK | Km bin. | 1mM | 08-180 | ||||||
BTK[C481S] | TK | Km bin. | 1mM | 08-547 | ||||||
BUB1/BUB3 | STK | Km bin. | Preincubation | 05-187 | ||||||
CaMK1α (CAMK1) | STK | Km bin. | 1mM | 02-104 | ||||||
CaMK1δ (CAMK1D) | STK | Km bin. | 02-106 | |||||||
CaMK2α (CAMK2A) | STK | Km bin. | Preincubation | 02-109 | ||||||
CaMK2β (CAMK2B) | STK | Km bin. | Preincubation | 02-110 | ||||||
CaMK2γ (CAMK2G) | STK | Km bin. | Preincubation | 02-112 | ||||||
CaMK2δ (CAMK2D) | STK | Km bin. | Preincubation | 02-111 | ||||||
CaMK4 | STK | Km bin. | 1mM | Preincubation | STK | 02-108 | ||||
CDC2/CycB1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-102 | ||||
CDC7/ASK | STK | Km bin. | 1mM | Cell Cycle | 05-109 | |||||
CDK2/CycA2 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 04-103 | |||
CDK2/CycE1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-165 | ||||
CDK3/CycE1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-104 | ||||
CDK4/CycD3 | STK | Km bin. | 1mM | Cell Cycle | 04-105 | |||||
CDK5/p25 | STK | Km bin. | 1mM | Preincubation | 04-106 | |||||
CDK6/CycD3 | STK | Km bin. | 1mM | Cell Cycle | 04-107 | |||||
CDK7/CycH/MAT1 | STK | Km bin. | 1mM | Cell Cycle | 04-108 | |||||
CDK9/CycT1 | STK | Km bin. | 1mM | Cell Cycle | 04-110 | |||||
CGK2 (PRKG2) | STK | Km bin. | Preincubation | 01-143 | ||||||
CHK1 (CHEK1) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 02-117 | |||
CHK2 (CHEK2) | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 02-162 | ||||
CK1α (CSNK1A1) | STK | Km bin. | 1mM | 03-101 | ||||||
CK1γ2 (CSNK1G1) | STK | Km bin. | Preincubation | 03-105 | ||||||
CK1γ2 (CSNK1G2) | STK | Km bin. | Preincubation | 03-106 | ||||||
CK1γ3 (CSNK1G3) | STK | Km bin. | Preincubation | 03-107 | ||||||
CK1δ (CSNK1D) | STK | Km bin. | Preincubation | 03-103 | ||||||
CK1ε (CSNK1E) | STK | Km bin. | 1mM | STK | 03-104 | |||||
CK2α1/β (CSNK2A1/B) | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 05-184 | ||||
CK2α2/β (CSNK2A2/B) | STK | Km bin. | Preincubation | Cell Cycle | 05-185 | |||||
CLK1 | STK | Km bin. | 1mM | Preincubation | 04-126 | |||||
CLK2 | STK | Km bin. | 1mM | Preincubation | 04-127 | |||||
CLK3 | STK | Km bin. | Preincubation | 04-128 | ||||||
COT (MAP3K8) | STK | 1mM (Cascade) | MAPK (Cascade) | 07-301 | ||||||
CRIK (CIT) | STK | Km bin. | 01-104 | |||||||
CSK | TK | Km bin. | 1mM | TK | 08-111 | |||||
DAPK1 | STK | Km bin. | 1mM | Preincubation | STK | 02-134 | ||||
DCAMKL2 | STK | Km bin. | 02-140 | |||||||
DDR1 | TK | Km bin. | 1mM | 08-113 | ||||||
DDR2 | TK | Km bin. | 1mM | 08-114 | ||||||
DLK (MAP3K12) | STK | 1mM (Cascade) | MAPK (Cascade) | 09-111 | ||||||
DYRK1A | STK | Km bin. | 1mM | Preincubation | 04-130 | |||||
DYRK1B | STK | Km bin. | 1mM | Preincubation | STK | 04-131 | ||||
DYRK2 | STK | Km bin. | Preincubation | 04-132 | ||||||
DYRK3 | STK | Km bin. | Preincubation | 04-133 | ||||||
EEF2K | STK | Km bin. | 10-113 | |||||||
EGFR | TK | Km bin. | 1mM | Preincubation | TK | 08-115 | ||||
EGFR[d746-750/T790M] | TK | Km bin. | 1mM | Preincubation | 08-528 | |||||
EGFR[d746-750] | TK | Km bin. | 1mM | Preincubation | 08-527 | |||||
EGFR[L858R] | TK | Km bin. | 1mM | Preincubation | 08-502 | |||||
EGFR[L861Q] | TK | Km bin. | 1mM | Preincubation | 08-513 | |||||
EGFR[T790M/L858R] | TK | Km bin. | 1mM | Preincubation | 08-510 | |||||
EGFR[T790M] | TK | Km bin. | 1mM | Preincubation | 08-194 | |||||
EML4-ALK | TK | Km bin. | 1mM | 08-516 | ||||||
EPHA1 | TK | Km bin. | 1mM | Preincubation | 08-119 | |||||
EPHA2 | TK | Km bin. | 1mM | Preincubation | TK | 08-121 | ||||
EPHA3 | TK | Km bin. | 1mM | Preincubation | 08-122 | |||||
EPHA4 | TK | Km bin. | 1mM | Preincubation | 08-123 | |||||
EPHA5 | TK | Km bin. | 1mM | Preincubation | 08-124 | |||||
EPHA6 | TK | Km bin. | 1mM | Preincubation | 08-125 | |||||
EPHA7 | TK | Km bin. | 1mM | Preincubation | 08-126 | |||||
EPHA8 | TK | Km bin. | 1mM | Preincubation | 08-127 | |||||
EPHB1 | TK | Km bin. | 1mM | Preincubation | 08-128 | |||||
EPHB2 | TK | Km bin. | 1mM | Preincubation | 08-129 | |||||
EPHB3 | TK | Km bin. | 1mM | Preincubation | 08-130 | |||||
EPHB4 | TK | Km bin. | 1mM | Preincubation | TK | 08-131 | ||||
Erk1 (MAPK3) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-142 | ||||
Erk2 (MAPK1) | STK | Km bin. | 1mM | Preincubation | STK | MAPK (Cascade) | 04-143 | |||
Erk5 (MAPK7) | STK | Km bin. | 1mM | MAPK (Cascade) | 04-146 | |||||
FAK (PTK2) | TK | Km bin. | 1mM | 08-137 | ||||||
FER | TK | Km bin. | 1mM | Preincubation | 08-139 | |||||
FES | TK | Km bin. | 1mM | Preincubation | 08-140 | |||||
FGFR1 | TK | Km bin. | 1mM | Preincubation | TK | 08-133 | ||||
FGFR1[V561M] | TK | Km bin. | 1mM | 08-536 | ||||||
FGFR2 | TK | Km bin. | 1mM | Preincubation | 08-134 | |||||
FGFR2[V564I] | TK | Km bin. | 1mM | Preincubation | 08-546 | |||||
FGFR3 | TK | Km bin. | 1mM | 08-135 | ||||||
FGFR3[K650E] | TK | Km bin. | 1mM | 08-501 | ||||||
FGFR3[K650M] | TK | Km bin. | 1mM | 08-199 | ||||||
FGFR3[V555L] | TK | Km bin. | 1mM | 08-548 | ||||||
FGFR3[V555M] | TK | Km bin. | 1mM | 08-543 | ||||||
FGFR4 | TK | Km bin. | 1mM | Preincubation | 08-136 | |||||
FGFR4[N535K] | TK | Km bin. | 1mM | 08-524 | ||||||
FGFR4[V550E] | TK | Km bin. | 1mM | 08-525 | ||||||
FGFR4[V550L] | TK | Km bin. | 1mM | Preincubation | 08-526 | |||||
FGR | TK | Km bin. | 1mM | Preincubation | 08-166 | |||||
FLT1 | TK | Km bin. | 1mM | Preincubation | 08-189 | |||||
FLT3 | TK | Km bin. | 1mM | TK | 08-154 | |||||
FLT4 | TK | Km bin. | 1mM | Preincubation | 08-190 | |||||
FMS (CSF1R) | TK | Km bin. | 1mM | 08-155 | ||||||
FRK | TK | Km bin. | 1mM | Preincubation | 08-167 | |||||
FYN [isoform a] | TK | Km bin. | 1mM | 08-168 | ||||||
FYN [isoform b] | TK | Km bin. | 1mM | 08-531 | ||||||
GSK3α (GSK3A) | STK | Km bin. | 1mM | Preincubation | 04-140 | |||||
GSK3β (GSK3B) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 04-141 | |||
Haspin (GSG2) | STK | Km bin. | Preincubation | 05-111 | ||||||
HCK | TK | Km bin. | 1mM | 08-169 | ||||||
HER2 | TK | Km bin. | 1mM | 08-016 | ||||||
HER4 (ERBB4) | TK | Km bin. | 1mM | Preincubation | 08-118 | |||||
HGK (MAP4K4) | STK | Km bin. | 1mM | STK | 07-137 | |||||
HIPK1 | STK | Km bin. | Preincubation | 04-135 | ||||||
HIPK2 | STK | Km bin. | Preincubation | 04-136 | ||||||
HIPK3 | STK | Km bin. | Preincubation | 04-137 | ||||||
HIPK4 | STK | Km bin. | 1mM | Preincubation | 04-138 | |||||
HPK1(MAP4K1) | STK | Km bin. | 07-410 | |||||||
IGF1R | TK | Km bin. | 1mM | Preincubation | TK | 08-141 | ||||
IKKα (CHUK) | STK | Km bin. | 05-112 | |||||||
IKKβ (IKBKB) | STK | Km bin. | 1mM | Preincubation | STK | 05-084 | ||||
IKKε (IKBKE) | STK | Km bin. | 05-114 | |||||||
INSR | TK | Km bin. | 1mM | Preincubation | 08-142 | |||||
IRAK1 | STK | Km bin. | 09-101 | |||||||
IRAK4 | STK | Km bin. | 1mM | STK | 09-145 | |||||
IRR (INSRR) | TK | Km bin. | 1mM | 08-143 | ||||||
ITK | TK | Km bin. | 1mM | TK | 08-181 | |||||
JAK1 | TK | Km bin. | 1mM | 08-144 | ||||||
JAK2 | TK | Km bin. | 1mM | Preincubation | 08-045 | |||||
JAK3 | TK | Km bin. | 1mM | Preincubation | TK | 08-046 | ||||
JNK1 (MAPK8) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-163 | ||||
JNK2 (MAPK9) | STK | Km bin. | 1mM | Preincubation | STK | MAPK (Cascade) | 04-164 | |||
JNK3 (MAPK10) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-150 | ||||
KDR | TK | Km bin. | 1mM | Preincubation | TK | 08-191 | ||||
KIT | TK | Km bin. | 1mM | 08-156 | ||||||
KIT[D816E] | TK | Km bin. | 1mM | 08-541 | ||||||
KIT[D816V] | TK | Km bin. | 1mM | 08-505 | ||||||
KIT[D816Y] | TK | Km bin. | 1mM | 08-534 | ||||||
KIT[T670I] | TK | Km bin. | 1mM | 08-195 | ||||||
KIT[V560G] | TK | Km bin. | 1mM | 08-504 | ||||||
KIT[V654A] | TK | Km bin. | 1mM | 08-511 | ||||||
LATS2 | STK | Km bin. | 01-124 | |||||||
LCK | TK | Km bin. | 1mM | Preincubation | TK | 08-170 | ||||
LOK (STK10) | STK | Km bin. | 07-315 | |||||||
LTK | TK | Km bin. | 1mM | 08-106 | ||||||
LYNa | TK | Km bin. | 1mM | Preincubation | 08-171 | |||||
LYNb | TK | Km bin. | 1mM | Preincubation | 08-172 | |||||
MAP2K1 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-141 | ||||||
MAP2K2 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-142 | ||||||
MAP2K3 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-143 | ||||||
MAP2K4 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-144 | ||||||
MAP2K5 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-145 | ||||||
MAP2K6 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-146 | ||||||
MAP2K7 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-148 | ||||||
MAP3K1 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-103 | ||||||
MAP3K2 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-104 | ||||||
MAP3K3 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-105 | ||||||
MAP3K4 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-106 | ||||||
MAP3K5 | STK | 1mM (Cascade) | MAPK (Cascade) | 07-107 | ||||||
MAP4K2 | STK | Km bin. | 07-111 | |||||||
MAPKAPK2 | STK | Km bin. | 1mM | Preincubation | STK | 02-142 | ||||
MAPKAPK3 | STK | Km bin. | Preincubation | 02-143 | ||||||
MAPKAPK5 | STK | Km bin. | Preincubation | 02-144 | ||||||
MARK1 | STK | Km bin. | Preincubation | 02-120 | ||||||
MARK2 | STK | Km bin. | Preincubation | 02-121 | ||||||
MARK3 | STK | Km bin. | Preincubation | 02-122 | ||||||
MARK4 | STK | Km bin. | Preincubation | 02-123 | ||||||
MELK | STK | Km bin. | 02-124 | |||||||
MER (MERTK) | TK | Km bin. | 1mM | Preincubation | 08-108 | |||||
MET | TK | Km bin. | 1mM | Preincubation | TK | 08-151 | ||||
MET[D1228H] | TK | Km bin. | 1mM | Preincubation | 08-540 | |||||
MET[M1250T] | TK | Km bin. | 1mM | Preincubation | 08-545 | |||||
MET [Y1235D] | TK | Km bin. | 1mM | Preincubation | 08-198 | |||||
MINK (MINK1) | STK | Km bin. | 1mM | 07-139 | ||||||
MLK1 (MAP3K9) | STK | 1mM (Cascade) | MAPK (Cascade) | 09-115 | ||||||
MLK2 (MAP3K10) | STK | 1mM (Cascade) | MAPK (Cascade) | 09-116 | ||||||
MLK3 (MAP3K11) | STK | 1mM (Cascade) | MAPK (Cascade) | 09-017 | ||||||
MNK1 (MKNK1) | STK | Km bin. | Preincubation | 02-145 | ||||||
MNK2 (MKNK2) | STK | Km bin. | Preincubation | 02-146 | ||||||
MOS | STK | 1mM (Cascade) | MAPK (Cascade) | 05-118 | ||||||
MRCKα (CDC42BPA) | STK | Km bin. | 01-107 | |||||||
MRCKβ (CDC42BPB) | STK | Km bin. | 01-108 | |||||||
MSK1 (RPS6KA5) | STK | Km bin. | Preincubation | 01-147 | ||||||
MSK2 (RPS6KA4) | STK | Km bin. | 01-148 | |||||||
MSSK1 (STK23) | STK | Km bin. | 04-159 | |||||||
MST1 (STK4) | STK | Km bin. | 1mM | STK | 07-116 | |||||
MST2 (STK3) | STK | Km bin. | 07-117 | |||||||
MST3 (STK24) | STK | Km bin. | 07-118 | |||||||
MST4 | STK | Km bin. | 07-119 | |||||||
MUSK | TK | Km bin. | 1mM | 08-153 | ||||||
NDR1 (STK38) | STK | Km bin. | 01-125 | |||||||
NDR2 (STK38L) | STK | Km bin. | 01-126 | |||||||
NEK1 | STK | Km bin. | 1mM | Cell Cycle | 05-123 | |||||
NEK2 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 05-226 | |||
NEK4 | STK | Km bin. | Preincubation | 05-128 | ||||||
NEK6 | STK | Km bin. | 1mM | Cell Cycle | 05-130 | |||||
NEK7 | STK | Km bin. | 1mM | Cell Cycle | 05-131 | |||||
NEK9 | STK | Km bin. | 1mM | Cell Cycle | 05-133 | |||||
NIM1K (MGC42105) | STK | Km bin. | Preincubation | 02-175 | ||||||
NPM1-ALK | TK | Km bin. | 1mM | Preincubation | 08-517 | |||||
NuaK1 | STK | Km bin. | Preincubation | 02-126 | ||||||
NuaK2 | STK | Km bin. | Preincubation | 02-127 | ||||||
p38α (MAPK14) | STK | Km bin. | 1mM | Preincubation | STK | MAPK (Cascade) | Cell Cycle | 04-152 | ||
p38β (MAPK11) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-153 | ||||
p38γ (MAPK12) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-155 | ||||
p38δ (MAPK13) | STK | Km bin. | 1mM | Preincubation | MAPK (Cascade) | 04-154 | ||||
p70S6K (RPS6KB1) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 01-154 | |||
p70S6Kβ (RPS6KB2) | STK | Km bin. | Preincubation | 01-155 | ||||||
PAK1 | STK | Km bin. | Preincubation | 07-123 | ||||||
PAK2 | STK | Km bin. | 1mM | Preincubation | STK | 07-124 | ||||
PAK4 | STK | Km bin. | 07-126 | |||||||
PAK5 (PAK7) | STK | Km bin. | Preincubation | 07-127 | ||||||
PAK6 | STK | Km bin. | 07-128 | |||||||
PASK | STK | Km bin. | 02-128 | |||||||
PBK | STK | Km bin. | 1mM | STK | 05-168 | |||||
PDGFRα (PDGFRA) | TK | Km bin. | 1mM | Preincubation | TK | 08-157 | ||||
PDGFRα (PDGFRA)[D842V] | TK | Km bin. | 1mM | Preincubation | 08-506 | |||||
PDGFRα (PDGFRA)[T674I] | TK | Km bin. | 1mM | 08-503 | ||||||
PDGFRα (PDGFRA)[V561D] | TK | Km bin. | 1mM | Preincubation | 08-507 | |||||
PDGFRβ (PDGFRB) | TK | Km bin. | 1mM | Preincubation | 08-158 | |||||
PDHK2 (PDK2) | STK | Km bin. | 10-140 | |||||||
PDHK4 (PDK4) | STK | Km bin. | 10-125 | |||||||
PDK1 (PDPK1) | STK | Km bin. | 1mM | STK | 01-132 | |||||
PEK (EIF2AK3) | STK | Km bin. | 05-155 | |||||||
PGK (PRKG1) | STK | Km bin. | 01-142 | |||||||
PHKG1 | STK | Km bin. | 02-152 | |||||||
PHKG2 | STK | Km bin. | 02-153 | |||||||
PIM1 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 02-054 | |||
PIM2 | STK | Km bin. | 1mM | Cell Cycle | 02-155 | |||||
PIM3 | STK | Km bin. | 02-156 | |||||||
PKACα (PRKACA) | STK | Km bin. | 1mM | STK | 01-127 | |||||
PKACβ (PRKACB) | STK | Km bin. | 01-128 | |||||||
PKACγ (PRKACG) | STK | Km bin. | 01-129 | |||||||
PKCα (PRKCA) | STK | Km bin. | 1mM | STK | 01-133 | |||||
PKCβ1 (PRKCB1) | STK | Km bin. | 01-134 | |||||||
PKCβ2 (PRKCB2) | STK | Km bin. | 01-165 | |||||||
PKCγ (PRKCG) | STK | Km bin. | 01-137 | |||||||
PKCδ (PRKCD) | STK | Km bin. | Preincubation | 01-135 | ||||||
PKCε (PRKCE) | STK | Km bin. | 1mM | Preincubation | 01-136 | |||||
PKCζ (PRKCZ) | STK | Km bin. | Preincubation | 01-141 | ||||||
PKCη (PRKCH) | STK | Km bin. | Preincubation | 01-138 | ||||||
PKCθ (PRKCQ) | STK | Km bin. | 01-140 | |||||||
PKCι (PRKCI) | STK | Km bin. | 01-139 | |||||||
PKD1 (PRKD1) | STK | Km bin. | Preincubation | 02-157 | ||||||
PKD2 (PRKD2) | STK | Km bin. | 1mM | Preincubation | STK | 02-158 | ||||
PKD3 (PRKD3) | STK | Km bin. | 02-159 | |||||||
PKN1 | STK | Km bin. | 01-144 | |||||||
PKR (EIF2AK2) | STK | Km bin. | 05-156 | |||||||
PLK1 | STK | Km bin. | 1mM | Cell Cycle | 05-157 | |||||
PLK2 | STK | Km bin. | Cell Cycle | 05-158 | ||||||
PLK3 | STK | Km bin. | 1mM | 05-159 | ||||||
PRKX | STK | Km bin. | 01-130 | |||||||
PYK2 (PTK2B) | TK | Km bin. | 1mM | Preincubation | TK | 08-138 | ||||
QIK (SNF1LK2) | STK | Km bin. | 1mM | Preincubation | 02-129 | |||||
RAF1 | STK | 1mM (Cascade) | MAPK (Cascade) | 09-125 | ||||||
RET | TK | Km bin. | 1mM | Preincubation | 08-159 | |||||
RET[G691S] | TK | Km bin. | 1mM | Preincubation | 08-522 | |||||
RET[M918T] | TK | Km bin. | 1mM | Preincubation | 08-508 | |||||
RET[S891A] | TK | Km bin. | 1mM | Preincubation | 08-523 | |||||
RET[Y791F] | TK | Km bin. | 1mM | Preincubation | 08-521 | |||||
ROCK1 | STK | Km bin. | 1mM | STK | 01-109 | |||||
ROCK2 | STK | Km bin. | Preincubation | 01-110 | ||||||
RON (MST1R) | TK | Km bin. | 1mM | Preincubation | 08-152 | |||||
ROS (ROS1) | TK | Km bin. | 1mM | Preincubation | 08-163 | |||||
RSK1(RPS6KA1) | STK | Km bin. | 1mM | Cell Cycle | 01-149 | |||||
RSK2 (RPS6KA3) | STK | Km bin. | Preincubation | 01-150 | ||||||
RSK3 (RPS6KA2) | STK | Km bin. | 1mM | Preincubation | 01-151 | |||||
RSK4 (RPS6KA6) | STK | Km bin. | 1mM | Preincubation | 01-152 | |||||
SGK | STK | Km bin. | 1mM | Preincubation | STK | 01-158 | ||||
SGK2 | STK | Km bin. | 01-159 | |||||||
SGK3SGKL | STK | Km bin. | Preincubation | 01-160 | ||||||
SIK (SNF1LK) | STK | Km bin. | 1mM | 02-131 | ||||||
skMLCK (MYLK2) | STK | Km bin. | 1mM | Preincubation | 02-150 | |||||
SLK | STK | Km bin. | 07-129 | |||||||
SPHK1 | Lipid | Km bin. | Preincubation | 11-105 | ||||||
SPHK2 | Lipid | Km bin. | 11-106 | |||||||
SRC | TK | Km bin. | 1mM | Preincubation | TK | 08-173 | ||||
SRM (SRMS) | TK | Km bin. | 1mM | Preincubation | 08-174 | |||||
SRPK1 | STK | Km bin. | 04-160 | |||||||
SRPK2 | STK | Km bin. | 04-161 | |||||||
SYK | TK | Km bin. | 1mM | TK | 08-176 | |||||
TAK1-TAB1 (MAP3K7) | STK | 1mM (Cascade) | MAPK (Cascade) | 09-019 | ||||||
TAOK2 | STK | Km bin. | 07-133 | |||||||
TBK1 | STK | Km bin. | Preincubation | 05-115 | ||||||
TEC | TK | Km bin. | 1mM | Preincubation | 08-182 | |||||
TIE2 (TEK) | TK | Km bin. | 1mM | Preincubation | TK | 08-185 | ||||
TNIK | STK | Km bin. | 1mM | 07-138 | ||||||
TNK1 | TK | Km bin. | 1mM | 08-104 | ||||||
TRKA (NTRK1) | TK | Km bin. | 1mM | TK | 08-186 | |||||
TRKB (NTRK2) | TK | Km bin. | 1mM | Preincubation | 08-187 | |||||
TRKC (NTRK3) | TK | Km bin. | 1mM | Preincubation | 08-197 | |||||
TSSK1 | STK | Km bin. | 1mM | Preincubation | STK | 02-364 | ||||
TSSK2 | STK | Km bin. | 02-165 | |||||||
TSSK3 | STK | Km bin. | 02-166 | |||||||
TXK | TK | Km bin. | 1mM | 08-183 | ||||||
TYK2 | TK | Km bin. | 1mM | 08-147 | ||||||
TYRO3 | TK | Km bin. | 1mM | Preincubation | TK | 08-109 | ||||
WNK1 | STK | Km bin. | 05-179 | |||||||
WNK2 | STK | Km bin. | 05-180 | |||||||
WNK3 | STK | Km bin. | 05-181 | |||||||
YESYES1 | TK | Km bin. | 1mM | Preincubation | 08-175 | |||||
YES(YES1)[T348I] | TK | Km bin. | 1mM | Preincubation | 08-533 | |||||
ZAP70 | TK | Km bin. | 1mM | 08-177 |